Palladium-catalyzed asymmetric sequential hydroalkylation and hydroamination of 1,3-enynes with 3-hydroxyindoles
Qiuyu Li, Ruixue Wu, Tao Wu, Renkang Wei, Zhijiao Li, Shang Gao, Minyan Wang, Hequan Yao, Aijun Lin
原始摘要（英文原文）· Original abstract
An unprecedented Pd-catalyzed asymmetric sequential hydroalkylation/hydroamination of 1,3-enynes was developed. This method provides efficient access to chiral pyrido[1,2- a ]indoles and derivatives in good yields with excellent enantioselectivities.