科研速览 · Science Skim继续刷下去 · Keep skimming →
◇ bioRxiv2026-09-12· bioinformatics

CRISPR-enhanced assessment of variants of unknown significance nominates oncology therapeutic targets and drug repositioning opportunities

A. Savino, A. Oikonomou, F. Perrone, R. R. De Lucia, L. De Pietri, Y. Belattar, L. Brown, M. L. Grau, K. McCarten, H. Najgebauer, U. Perron, L. Azzolin, A. Livanova, P. Cremaschi, N. Lopez-Bigas, A. Sottoriva, M. A. Coelho, F. IORIO

原始摘要(英文原文)· Original abstract
Interpreting infrequent somatic variants remains a challenge in cancer genomics. We developed CRISPR-VUS, a framework that uses public Cancer Dependency Map data to identify Dependency-Associated Mutations (DAMs) - variants linked to increased host-gene dependency - with resolution extending to singleton events. Analysis of 977 cell lines across 36 cancer types identified 2,376 DAMs in 1,383 genes, including 1,260 not established as cancer drivers. DAM-bearing genes converge on oncogenic networks, while recurrence in histology-matched tumours, functional-impact predictions, tractability and pharmacological associations enable systematic prioritisation. Prime editing showed that the prioritised NSCLC-specific RTN4IP1-A80T DAM conferred a significant competitive growth advantage in a lung epithelial model, nominating a candidate driver allele. Exploratory pharmacological testing showed a greater maximal response to istaroxime in ATP1B3-I189M-bearing than in ATP1B3-wild-type cells. CRISPR-VUS combines dependency-based rare-variant discovery with evidence-guided prioritisation to nominate candidate drivers, therapeutic targets and drug-repositioning hypotheses. Interactive results are available at https://vus-portal.fht.org/.
读原文 · Read the paper ↗

AI 追问PRO

登录后使用 AI 追问

讨论区

登录后参与讨论

相关论文 · Related

CRISPR-enhanced assessment of variants of unknown significance nominates oncology therapeutic targets and drug repositioning opportunities — 科研速览 Science Skim