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◆ Biomaterials Science2026-01-01· Cytosol

Glutathione-activatable bola dendrimers mediate tumor-specific cytosolic siRNA delivery <i>via</i> dynamic thiol–disulfide exchange

Dandan Zhu, Huiling Zhu, Yaoyun Yu, Junyue Zheng, Xianhui Lin, Huimin Cheng, Aoxue Mei, Ming Chen, Yun Li, Haijuan Dong, Jiehua Zhou, Juan LIU, Xiaoxuan Liu

原始摘要(英文原文)· Original abstract
achieved substantial reductions in tumor growth and PLK1 expression while exhibiting minimal systemic toxicity. This study highlights a synergistic approach utilizing bola-amphiphilic peptide dendrimers for tumor-specific and cytosolic siRNA delivery, leveraging membrane-thiol interactions and intracellular GSH-triggered siRNA release.
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Glutathione-activatable bola dendrimers mediate tumor-specific cytosolic siRNA delivery <i>via</i> dynamic thiol–disulfide exchange — 科研速览 Science Skim