Rapid Microwave‐Assisted Iodination of Glycals to 2‐Iodoglycals Under Operationally Simple Conditions: Next Chapter in (C‐2)‐Functionalisation of Sugar Moieties
Dariusz Baran, Agnieszka Ewa Kuklewska, Morgane de Robichon, Bartłomiej Stankiewicz, Karolina Hurej, Aneta Pobudkowska, Andrzej Plichta, Angélique Ferry, Maciej Malinowski
原始摘要(英文原文)· Original abstract
Herein, we report an improved, microwave‐assisted protocol towards 2‐iodoglycals. The procedure itself is efficient, easy to reproduce and might be transferred onto challenging examples of glycals, such as trisaccharide derivatives or analogues of antidiabetic acarbose allowing the synthesis of their 2‐iodoanalogues in few minutes.
Rapid Microwave‐Assisted Iodination of Glycals to 2‐Iodoglycals Under Operationally Simple Conditions: Next Chapter in (C‐2)‐Functionalisation of Sugar Moieties — 科研速览 Science Skim